Development of a new cascade reaction for convergent synthesis of pyrazolo[1,5-a]quinoline derivatives under transition-metal-free conditions.

نویسندگان

  • Jun-ya Kato
  • Hiroshi Aoyama
  • Tsutomu Yokomatsu
چکیده

A novel method for the synthesis of pyrazolo[1,5-a]quinolines under the transition-metal-free conditions has been developed. This method involves a novel combination of aromatic nucleophilic substitution and Knoevenagel condensation reactions to give pyrazolo[1,5-a]quinolines.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 11 7  شماره 

صفحات  -

تاریخ انتشار 2013